1. Signaling Pathways
  2. Vitamin D Related/Nuclear Receptor
  3. Estrogen Receptor/ERR
  4. Estrogen receptor Isoform
  5. Estrogen receptor Inhibitor

Estrogen receptor Inhibitor

Estrogen receptor Inhibitors (2):

Cat. No. Product Name Effect Purity
  • HY-135309
    PROTAC ER Degrader-4
    Inhibitor 98.22%
    PROTAC ER Degrader-4 is a von Hippel-Lindau-based PROATC estrogen receptor (ER) degrader, binding to ER with an IC50 of 0.8 nM. PROTAC ER Degrader-4 induces ER degradation in MCF-7 cells with an IC50 of 0.3 nM.
  • HY-113251
    2-Hydroxyestrone
    Inhibitor 98.57%
    2-Hydroxyestrone (Catecholestrone) is a specific receptor-mediated antiestrogenic agent. 2-Hydroxyestrone is anticarcinogenic.